SCHEMBL8005538

SCHEMBL8005538

COC(=O)Cc1ccc(Oc2ccc3c(c2)COB3)c(F)c1

nearest known ligand 0.41

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.41
ROCK1 Q13464 1/20 0.41
MMP9 P14780 1/20 0.38
LMNA P02545 1/20 0.36
FFAR1 O14842 3/20 0.36
ALDH1A1 P00352 2/20 0.36
GAA P10253 1/20 0.36
GFER P55789 1/20 0.36
MAPK14 Q16539 1/20 0.35
PPARD Q03181 1/20 0.35
MAPT P10636 1/20 0.34
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
LIPE Q05469 1/20 0.34
OPRM1 P35372 1/20 0.34
OPRD1 P41143 1/20 0.34
OPRK1 P41145 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006261 0.87 MMP9 (0.36) MMP9LMNAFFAR1ALDH1A1GAA
SCHEMBL16472180 0.83 USP2 (0.40) LMNAALDH1A1MAPK14MAPTHPGD
SCHEMBL14748412 0.78 PDE4B (0.41) GAAMAPTOPRM1OPRD1OPRK1
SCHEMBL8006270 0.77 KMT2A (0.41) MMP9ALDH1A1HPGDTSHR
SCHEMBL16870235 0.76 PPARD (0.47) ROCK2LMNAALDH1A1GAAGFER
SCHEMBL8007014 0.75 MMP9 (0.37) ROCK2ROCK1MMP9LMNAALDH1A1
SCHEMBL8008270 0.74 LMNA (0.54) LMNAALDH1A1MAPTTSHRLIPE
SCHEMBL1039522 0.72 HTT (0.51) LMNAALDH1A1GAAGFERHPGD
SCHEMBL4843750 0.69 ALDH1A1 (0.49) LMNAALDH1A1GAAGFER
SCHEMBL7997146 0.69 PTGDR2 (0.42) FFAR1PPARDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111676-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS ANACOR PHARMACEUTICALS, INC (US) 2009-09-11 WO disclosed