SCHEMBL8007014

SCHEMBL8007014

COC(=O)Cc1ccc(Oc2ccc3c(c2)COB3)cc1Cl

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 2/20 0.37
ALDH1A1 P00352 4/20 0.37
HTT P42858 2/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
THRB P10828 1/20 0.37
LMNA P02545 1/20 0.35
KDM4E B2RXH2 3/20 0.35
HPGD P15428 1/20 0.35
ROCK2 O75116 1/20 0.34
ROCK1 Q13464 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
RET P07949 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
SLC5A1 P13866 1/20 0.33
SLC5A2 P31639 1/20 0.33
PDE4A P27815 3/20 0.33
PDE4B Q07343 3/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8006270 0.86 KMT2A (0.41) MMP9ALDH1A1MEN1KMT2AKDM4E
SCHEMBL8008270 0.79 LMNA (0.54) ALDH1A1LMNANPC1RAB9AMAPT
SCHEMBL8006261 0.76 MMP9 (0.36) MMP9ALDH1A1THRBLMNAHPGD
SCHEMBL8005538 0.75 ROCK2 (0.41) MMP9ALDH1A1LMNAHPGDROCK2
SCHEMBL473984 0.74 ALDH1A1 (0.53) ALDH1A1HTTL3MBTL1MEN1KMT2A
SCHEMBL14748434 0.72 PDE4A (0.50) ALDH1A1HTTL3MBTL1MEN1KMT2A
SCHEMBL5801556 0.70 PDE4A (0.49) PDE4APDE4BPDE4CPDE4D
SCHEMBL8007094 0.69 PDE4A (0.50) MMP9PDE4APDE4BPDE4CPDE4D
SCHEMBL19622266 0.69 ALDH1A1 (0.47) ALDH1A1MEN1KMT2ALMNAHPGD
SCHEMBL837451 0.68 ALDH1A1 (0.56) ALDH1A1HTTL3MBTL1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111676-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS ANACOR PHARMACEUTICALS, INC (US) 2009-09-11 WO disclosed