SCHEMBL8006261

SCHEMBL8006261

COC(=O)Cc1cc(F)c(Oc2ccc3c(c2)COB3)c(F)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP9 P14780 1/20 0.36
HSP90AB1 P08238 1/20 0.36
LMNA P02545 1/20 0.35
LIPE Q05469 1/20 0.33
ALDH1A1 P00352 2/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
GAA P10253 1/20 0.32
GFER P55789 1/20 0.32
CYP4F2 P78329 1/20 0.32
CYP4A11 Q02928 1/20 0.32
PCNA P12004 2/20 0.32
FFAR1 O14842 1/20 0.32
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
PDK2 Q15119 1/20 0.31
MAPT P10636 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8005538 0.87 ROCK2 (0.41) MMP9LMNALIPEALDH1A1NPC1
SCHEMBL14748413 0.79 PDE4B (0.40) LMNAALDH1A1GAAMAPTHPGD
SCHEMBL8006270 0.76 KMT2A (0.41) MMP9ALDH1A1HPGDTSHR
SCHEMBL8007014 0.76 MMP9 (0.37) MMP9LMNAALDH1A1NPC1RAB9A
SCHEMBL8008270 0.76 LMNA (0.54) LMNALIPEALDH1A1NPC1RAB9A
SCHEMBL8007094 0.71 PDE4A (0.50) MMP9MAOB
SCHEMBL8012386 0.70 PDE4B (0.34) ALDH1A1HPGD
SCHEMBL19622171 0.69 TSHR (0.54) LMNAALDH1A1GAAMAPTHPGD
SCHEMBL2126802 0.69 HSP90AB1 (0.56) HSP90AB1ALDH1A1GAAGFERCYP4F2
SCHEMBL8010793 0.68 ST14 (0.51) MMP9MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009111676-A2 BORON-CONTAINING SMALL MOLECULES AS ANTI-INFLAMMATORY AGENTS ANACOR PHARMACEUTICALS, INC (US) 2009-09-11 WO disclosed