SCHEMBL8010267

SCHEMBL8010267

Cc1nc(C(C)(C)C/C=C/c2cccc(-c3nn(C)nc3-c3ccccc3)c2)cs1

nearest known ligand 0.33

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 8/20 0.33
HDAC8 Q9BY41 8/20 0.33
HDAC6 Q9UBN7 8/20 0.33
ALDH1A1 P00352 2/20 0.31
HPGD P15428 2/20 0.31
KDM4E B2RXH2 1/20 0.31
HSD17B10 Q99714 1/20 0.31
RXFP1 Q9HBX9 1/20 0.31
GRM5 P41594 1/20 0.31
HTT P42858 1/20 0.30
PTGS2 P35354 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7998518 0.85 PKM (0.33) HDAC1HDAC8HDAC6ALDH1A1HPGD
SCHEMBL7998466 0.81 PKM (0.36) HDAC1HDAC8HDAC6ALDH1A1HPGD
SCHEMBL7998514 0.80 PKM (0.38) HDAC1HDAC8HDAC6ALDH1A1HPGD
SCHEMBL8000613 0.80 L3MBTL1 (0.32) ALDH1A1KDM4E
SCHEMBL7998465 0.80 PKM (0.39) HDAC1HDAC8HDAC6ALDH1A1HPGD
SCHEMBL10292921 0.79
SCHEMBL7998468 0.77 PKM (0.37) HDAC1HDAC8HDAC6ALDH1A1HTT
SCHEMBL7998573 0.77 PRMT6 (0.36) HDAC1HDAC8HDAC6ALDH1A1HPGD
SCHEMBL7998527 0.73 GRIN1 (0.35) HDAC1HDAC8HDAC6
SCHEMBL8007763 0.68 GRIN1 (0.35) HDAC1HDAC8HDAC6ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed