SCHEMBL7998466

SCHEMBL7998466

Cc1nc(C/C=C/c2cccc(-c3nn(C)nc3-c3ccccc3)c2)cs1

nearest known ligand 0.40

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.36
HDAC1 Q13547 5/20 0.35
HDAC8 Q9BY41 5/20 0.35
HDAC6 Q9UBN7 5/20 0.35
SLC6A3 Q01959 3/20 0.34
SLC12A2 P55011 1/20 0.34
SLC12A5 Q9H2X9 1/20 0.34
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 1/20 0.33
HSD17B10 Q99714 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
GRM5 P41594 1/20 0.33
USP2 O75604 1/20 0.33
ALOX15 P16050 1/20 0.33
MAPK1 P28482 1/20 0.33
MAPT P10636 1/20 0.32
DCTPP1 Q9H773 1/20 0.32
TSHR P16473 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7998465 0.89 PKM (0.39) PKMHDAC1HDAC8HDAC6SLC6A3
SCHEMBL7998514 0.88 PKM (0.38) PKMHDAC1HDAC8HDAC6SLC6A3
SCHEMBL7998518 0.87 PKM (0.33) PKMHDAC1HDAC8HDAC6SLC6A3
SCHEMBL7998468 0.87 PKM (0.37) PKMHDAC1HDAC8HDAC6SLC6A3
SCHEMBL8010267 0.81 HDAC1 (0.33) HDAC1HDAC8HDAC6ALDH1A1KDM4E
SCHEMBL7998537 0.78 L3MBTL1 (0.34) HDAC1HDAC8HDAC6SLC6A3SLC12A2
SCHEMBL10292927 0.77 SLC6A3 (0.36) SLC6A3
SCHEMBL10260889 0.77 SLC6A3 (0.36) SLC6A3
SCHEMBL8008282 0.76 PKM (0.42) PKMSLC6A3SLC12A2SLC12A5GRM5
SCHEMBL8007763 0.75 GRIN1 (0.35) HDAC1HDAC8HDAC6ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009134987-A1 DIFLUOROMETHYL-CONTAINING MACROCYCLIC COMPOUNDS AS HEPATITIS C VIRUS INHIBITORS ENANTA PHARMACEUTICALS, INC. (US) 2009-11-05 WO disclosed