SCHEMBL8015147

SCHEMBL8015147

C1=C(C2=CCNCC2)CCN1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 2/20 0.52
HTR2C P28335 8/20 0.50
QDPR P09417 2/20 0.48
HRH3 Q9Y5N1 1/20 0.44
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
MAPT P10636 1/20 0.40
DRD2 P14416 1/20 0.40
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40
GABRP O00591 1/20 0.38
GABRD O14764 1/20 0.38
GABRA1 P14867 1/20 0.38
TSHR P16473 1/20 0.38
GABRB1 P18505 1/20 0.38
GABRG2 P18507 1/20 0.38
GABRR1 P24046 1/20 0.38
GABRB3 P28472 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRA3 P34903 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21361657 0.73 SIGMAR1 (0.52) SIGMAR1HTR2CQDPRHRH3KDM4E
SCHEMBL3803151 0.71 HTR2C (0.47) SIGMAR1HTR2CQDPRHRH3
SCHEMBL11246723 0.71 SIGMAR1 (0.50) SIGMAR1HTR2CQDPRHRH3KDM4E
SCHEMBL24052807 0.69 SIGMAR1 (0.43) SIGMAR1HTR2CQDPRHRH3KDM4E
SCHEMBL918294 0.69 ADRA2A (0.31)
SCHEMBL415545 0.68 SIGMAR1 (1.00) SIGMAR1HTR2CQDPRKDM4EALDH1A1
SCHEMBL23074510 0.67 SIGMAR1 (0.46) SIGMAR1HTR2CQDPRHRH3KDM4E
SCHEMBL18372897 0.67
SCHEMBL5542927 0.67 HTR2C (0.50) SIGMAR1HTR2CQDPRHRH3KDM4E
Bromide SCHEMBL11385943 0.67 SIGMAR1 (0.96) SIGMAR1HTR2CQDPRKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0969842-A1 PHARMACEUTICAL COMPOSITION R.P. Scherer Limited (GB) 2000-01-12 EP disclosed
WO-1998042344-A1 PHARMACEUTICAL COMPOSITION R. P. SCHERER LIMITED (GB) 1998-10-01 WO disclosed