SCHEMBL801870

SCHEMBL801870

Cc1nc(Cl)nc(Cl)c1C

nearest known ligand 0.39

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.39
ALOX15 P16050 1/20 0.39
TSHR P16473 1/20 0.39
PDE10A Q9Y233 2/20 0.37
CYP1A2 P05177 1/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL812036 0.84 PDE10A (0.48) ALDH1A1ALOX15TSHRPDE10ACYP1A2
SCHEMBL1586433 0.84 ALDH1A1 (0.47) ALDH1A1ALOX15TSHRPDE10AMEN1
SCHEMBL1703281 0.77 LMNA (0.45) ALDH1A1ALOX15TSHRCYP1A2MEN1
SCHEMBL1830615 0.77 PDE10A (0.37) PDE10A
SCHEMBL6462055 0.74 MEN1 (0.39) ALDH1A1ALOX15TSHRMEN1KMT2A
SCHEMBL439985 0.73 PDE10A (0.39) PDE10A
SCHEMBL8382893 0.72 ALDH1A1 (0.30) ALDH1A1ALOX15TSHR
SCHEMBL23443915 0.72 ALDH1A1 (0.35) ALDH1A1ALOX15TSHR
SCHEMBL10043017 0.72 ALDH1A1 (0.35) ALDH1A1ALOX15TSHR
SCHEMBL10603143 0.72 PDE10A (0.52) ALDH1A1ALOX15TSHRPDE10A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 167 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260132147-A1 BAX INHIBITORS AND USES THEREOF CASE WESTERN RESERVE UNIV (US) 2026-05-14 US disclosed
US-12552790-B2 Positive modulators of the muscarinic acetylcholine receptor M4 VANDERBILT UNIVERSITY (US) 2026-02-17 US disclosed
US-20260035366-A1 POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 UNIV VANDERBILT (US) 2026-02-05 US disclosed
US-20260034127-A1 TREATMENT OF GVHD KADMON CORP LLC (FR) 2026-02-05 US disclosed
US-12479857-B2 Bax inhibitors and uses thereof CASE WESTERN RESERVE UNIVERSITY (US) 2025-11-25 US disclosed
US-12448380-B2 Positive modulators of the muscarinic acetylcholine receptor M4 VANDERBILT UNIVERSITY (US) 2025-10-21 US disclosed
US-20250230155-A1 7,8-DIHYDRO-5H-1,6-NAPHTHYRIDINE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS VANDERBILT UNIVERSITY 2025-07-17 US disclosed
US-12344608-B2 Positive modulators of the muscarinic acetylcholine receptor M4 VANDERBILT UNIVERSITY (US) 2025-07-01 US disclosed
US-20250136600-A1 POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY 2025-05-01 US disclosed
US-20250122198-A1 POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 VANDERBILT UNIVERSITY 2025-04-17 US disclosed
US-6545008-B1 Inhibitory activity against gastric acid secretion YUHAN CORPORATION (KR) 2003-04-08 US disclosed
US-6352993-B1 ANTIULCER AGENTS YUHAN CORPORATION (KR) 2002-03-05 US disclosed
CN-1326453-A Novel poyrimidine derivatives and process for preparation thereof YUHAN CORP (KR) 2001-12-12 CN disclosed
EP-1131312-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION, LTD. (KR) 2001-09-12 EP disclosed
WO-2000029403-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 2000-05-25 WO disclosed
US-5750531-A ANTISECRETORY AGENTS FOR THE TREATMENT OF PEPTIC ULCER YUHAN CORPORATION (KR) 1998-05-12 US disclosed
EP-0775120-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF Yuhan Corporation (KR) 1997-05-28 EP disclosed
WO-1996005177-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 1996-02-22 WO disclosed
US-4980350-A Piperazinylalkylpyrimidines as hypoglycemic agents MERCK & CO., INC. (US) 1990-12-25 US disclosed
EP-0330263-A1 Piperazinylalkylpyrimidines as hypoglycemic agents MERCK & CO. INC. (US) 1989-08-30 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260132147-A1 BAX INHIBITORS AND USES THEREOF BAX, BCL2, BAK1 ALDH1A1 4585/4885ALOX15 997/4885TSHR 3456/4885
US-12552790-B2 Positive modulators of the muscarinic acetylcholine receptor M4 CHRM4, CHRM1, CHRM5 ALDH1A1 2392/4885ALOX15 4512/4885TSHR 37/4885
US-20250136600-A1 POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 CHRM4, CHRM1, CHRM3 ALDH1A1 2993/4885ALOX15 4041/4885TSHR 51/4885
US-20260034127-A1 TREATMENT OF GVHD ROCK2, RHOA, MYH2 ALDH1A1 3146/4885ALOX15 4352/4885TSHR 4630/4885
US-12344608-B2 Positive modulators of the muscarinic acetylcholine receptor M4 CHRM4, CHRM1, CHRM3 ALDH1A1 2993/4885ALOX15 4041/4885TSHR 51/4885
US-20250122198-A1 POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 CHRM4, CHRM1, CHRM3 ALDH1A1 2993/4885ALOX15 4041/4885TSHR 51/4885
US-12479857-B2 Bax inhibitors and uses thereof BAX, TMBIM6, BCL2 ALDH1A1 4296/4885ALOX15 2696/4885TSHR 4763/4885
US-20260035366-A1 POSITIVE MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 CHRM4, CHRM3, CHRM5 ALDH1A1 3334/4885ALOX15 3943/4885TSHR 67/4885
US-20250230155-A1 7,8-DIHYDRO-5H-1,6-NAPHTHYRIDINE DERIVATIVES AS POSITIVE ALLOSTERIC MODULATORS OF THE MUSCARINIC ACETYLCHOLINE RECEPTOR M4 FOR TREATING NEUROLOGICAL AND PSYCHIATRIC DISORDERS CHRM5, CHRM4, CHRM1 ALDH1A1 1671/4885ALOX15 4659/4885TSHR 123/4885
US-12448380-B2 Positive modulators of the muscarinic acetylcholine receptor M4 CHRM4, CHRM1, CHRM3 ALDH1A1 2993/4885ALOX15 4041/4885TSHR 51/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.