SCHEMBL8018985

SCHEMBL8018985

CC(C)(C)OC(=O)N(C(=O)c1cccc(F)c1)C1CC1C(=O)O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.39
OPRL1 P41146 1/20 0.39
GRM5 P41594 2/20 0.38
KMT2A Q03164 3/20 0.36
MEN1 O00255 2/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
TSHR P16473 1/20 0.36
GAA P10253 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
PARP1 P09874 1/20 0.35
HTT P42858 2/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
ALDH1A1 P00352 2/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
POLB P06746 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
PIK3CD O00329 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8025166 0.86 GAA (0.42) GRM5KMT2AMEN1GAAL3MBTL1
SCHEMBL8018895 0.86 MEN1 (0.36) KMT2AMEN1TSHRGAAL3MBTL1
SCHEMBL8025266 0.85 TAS1R3 (0.37) KMT2AMEN1CES2CES1RAB9A
SCHEMBL8007793 0.73 CES2 (0.44) GRM5KMT2AMEN1CES2CES1
SCHEMBL4224819 0.68 ESR1 (0.55) KMT2AMEN1CES2CES1PARP1
SCHEMBL30437641 0.68 ESR1 (0.55) KMT2AMEN1CES2CES1PARP1
SCHEMBL25244239 0.67 CES2 (0.42) OPRM1OPRL1KMT2AMEN1CES2
SCHEMBL8008096 0.66 KMO (0.55) GRM5KMT2AMEN1CES2CES1
SCHEMBL12084828 0.66 CES2 (0.55) OPRM1OPRL1GRM5KMT2AMEN1
SCHEMBL6050410 0.65 CTNNB1 (0.42) KMT2AMEN1CES2CES1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973720-A1 2-SUBSTITUTED BENZOYL-CYCLOALKYL-1-CARBOXYLIC ACID DERIVATIVES PHARMACIA & UPJOHN S.p.A. (IT) 2000-01-26 EP disclosed
WO-1998040344-A1 2-SUBSTITUTED BENZOYL-CYCLOALKYL-1-CARBOXYLIC ACID DERIVATIVES PHARMACIA & UPJOHN S.P.A. (IT) 1998-09-17 WO disclosed