SCHEMBL8020531

SCHEMBL8020531

Fc1ccc(P(Cc2ccc3ccccc3c2-c2c(CP(c3ccc(F)cc3F)c3ccc(F)cc3F)ccc3ccccc23)c2ccc(F)cc2F)c(F)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.37
CYP1A2 P05177 1/20 0.37
MAPK14 Q16539 1/20 0.36
HPRT1 P00492 1/20 0.36
TRPA1 O75762 1/20 0.35
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
AHR P35869 1/20 0.32
PPARG P37231 1/20 0.32
IDO1 P14902 2/20 0.32
AGXT P21549 2/20 0.32
ALDH1A1 P00352 3/20 0.31
KDM4E B2RXH2 1/20 0.31
NPC1 O15118 1/20 0.31
GAA P10253 1/20 0.31
NFKB1 P19838 1/20 0.31
RAB9A P51151 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6423410 0.85 HPRT1 (0.38) CYP2A6CYP1A2HPRT1AHRALDH1A1
SCHEMBL8022927 0.85 HPRT1 (0.36) CYP2A6HPRT1AHRALDH1A1KDM4E
SCHEMBL8022208 0.79 CES1 (0.37) CYP2A6CYP1A2HPRT1ALDH1A1NPC1
SCHEMBL8010779 0.78 CYP1A2 (0.36) CYP2A6CYP1A2HPRT1AHRALDH1A1
SCHEMBL8023352 0.78 HPGD (0.35) CYP2A6CYP1A2HPRT1AHRALDH1A1
SCHEMBL6420832 0.78 CYP2A6 (0.36) CYP2A6CYP1A2HPRT1AHRALDH1A1
SCHEMBL8056031 0.77 CES1 (0.36) CYP2A6CYP1A2HPRT1ALDH1A1NPC1
SCHEMBL6418430 0.77 HPRT1 (0.38) CYP2A6CYP1A2HPRT1AHRALDH1A1
SCHEMBL6424099 0.74 ALDH1A1 (0.35) CYP2A6HPRT1ALDH1A1CES1HSD17B10
SCHEMBL8010374 0.73 CYP2A6 (0.41) CYP2A6CYP1A2ALDH1A1HSD17B10TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653432-B1 Process for preparing bis-(diaryl-alkyl)-phosphines and derivatives of this class of substances CELANESE CHEM EUROPE GMBH (DE) 2000-02-09 EP claimed
US-5600006-A Bis(diarylalkyl)phosphines HOECHST A.G. (DE) 1997-02-04 US claimed
EP-0653432-A1 Process for preparing bis-(diaryl-alkyl)-phosphines and novel derivatives of this class of substances HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-17 EP claimed
EP-0653432-B1 Process for preparing bis-(diaryl-alkyl)-phosphines and derivatives of this class of substances CELANESE CHEM EUROPE GMBH (DE) 2000-02-09 EP disclosed
US-5600006-A Bis(diarylalkyl)phosphines HOECHST A.G. (DE) 1997-02-04 US disclosed
EP-0653432-A1 Process for preparing bis-(diaryl-alkyl)-phosphines and novel derivatives of this class of substances HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-17 EP disclosed