SCHEMBL8024217

SCHEMBL8024217

COc1ccc(-c2ccc(CO)c(OC)c2)c(Cl)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDCD1 Q15116 2/20 0.56
CD274 Q9NZQ7 2/20 0.56
CYP11B1 P15538 1/20 0.45
CYP11B2 P19099 1/20 0.45
ERN1 O75460 1/20 0.44
PDE5A O76074 1/20 0.44
PDE4A P27815 1/20 0.44
PDE1A P54750 1/20 0.44
PDE1B Q01064 1/20 0.44
PDE4B Q07343 1/20 0.44
PDE4C Q08493 1/20 0.44
PDE4D Q08499 1/20 0.44
PDE3B Q13370 1/20 0.44
PDE1C Q14123 1/20 0.44
PDE3A Q14432 1/20 0.44
CYP1A2 P05177 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP1A1 P04798 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7945286 0.87 PDCD1 (0.43) PDCD1CD274CYP11B1CYP11B2ERN1
SCHEMBL7944717 0.86 CYP11B1 (0.45) PDCD1CD274CYP11B1CYP11B2CYP1A2
SCHEMBL8017441 0.84 PDCD1 (0.61) PDCD1CD274CYP11B1CYP11B2PDE5A
SCHEMBL8028294 0.80 PDCD1 (0.58) PDCD1CD274ERN1PDE5APDE4A
SCHEMBL4050630 0.80 PDCD1 (0.52) PDCD1CD274CYP11B1CYP11B2PDE5A
SCHEMBL238087 0.79 APLNR (0.63) PDCD1CD274PDE4APDE4BPDE4C
Methylene Chloride SCHEMBL28275708 0.78 APLNR (0.58) PDCD1CD274PDE4APDE4BPDE4C
SCHEMBL5753110 0.78 ALDH1A1 (0.54) CYP11B1CYP11B2APLNRKDM4EALDH1A1
SCHEMBL28303202 0.77 ESR2 (0.57) CYP1A2CYP3A4CYP2D6CYP2C19CYP1A1
SCHEMBL12325069 0.76 HSP90AA1 (0.56) CYP11B1CYP11B2CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009071504-A1 2,6-DISUBSTITUTED PYRIDINES AS SOLUBLE GUANYLATE CYCLASE ACTIVATORS SMITHKLINE BEECHAM CORPORATION (US) 2009-06-11 WO disclosed