SCHEMBL8024511

SCHEMBL8024511

O=C(O)CN(C(=O)C(CS)CCc1ccccc1)c1cccc(OCc2ccc(C(=O)O)cc2)c1

nearest known ligand 0.50

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
SRD5A2 P31213 2/20 0.47
NR4A2 P43354 5/20 0.46
ALOX5 P09917 3/20 0.46
PTGES O14684 2/20 0.46
LTC4S Q16873 1/20 0.46
RXRA P19793 1/20 0.45
RXRB P28702 1/20 0.45
RXRG P48443 1/20 0.45
FFAR1 O14842 2/20 0.43
NR4A1 P22736 1/20 0.43
NR4A3 Q92570 1/20 0.43
NR1H4 Q96RI1 1/20 0.41
PTGER1 P34995 1/20 0.41
PTGER4 P35408 1/20 0.41
PTGER3 P43115 1/20 0.41
PTGER2 P43116 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8022583 0.94 FFAR1 (0.46) SMN1; SMN2NR4A2ALOX5FFAR1
SCHEMBL8023084 0.93 MRGPRX4 (0.49) NR4A2FFAR1NR1H4
SCHEMBL8026747 0.90 ALOX5 (0.52) SMN1; SMN2SRD5A2NR4A2ALOX5PTGES
SCHEMBL8161868 0.85 ACE (0.41)
SCHEMBL8024336 0.84 FFAR1 (0.50) ALOX5FFAR1
SCHEMBL8023170 0.84 FFAR1 (0.42) FFAR1PTGER3
SCHEMBL8010560 0.84 MRGPRX4 (0.48) SMN1; SMN2NR4A2NR1H4
SCHEMBL8020340 0.83 MMP12 (0.48) ALOX5FFAR1
SCHEMBL8010235 0.82 MMP12 (0.47) ALOX5FFAR1
SCHEMBL8010404 0.80 FFAR1 (0.49) FFAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US claimed
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed