SCHEMBL8010235

SCHEMBL8010235

O=C(O)CN(C(=O)C(CS)CCc1ccccc1)c1ccc(OCc2ccc(O)cc2)cc1

nearest known ligand 0.66

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.47
FFAR1 O14842 5/20 0.47
FFAR4 Q5NUL3 2/20 0.47
MAOB P27338 2/20 0.45
LMNA P02545 1/20 0.45
CYP1A2 P05177 1/20 0.45
PTGS1 P23219 1/20 0.45
SLC6A2 P23975 1/20 0.45
CYP2C19 P33261 1/20 0.45
PTGS2 P35354 1/20 0.45
SLC6A3 Q01959 1/20 0.45
HIF1A Q16665 1/20 0.45
HDAC6 Q9UBN7 1/20 0.45
KEAP1 Q14145 1/20 0.43
BCHE P06276 1/20 0.43
ALOX5 P09917 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8024336 0.97 FFAR1 (0.50) MMP12FFAR1FFAR4MAOBKEAP1
SCHEMBL8020340 0.96 MMP12 (0.48) MMP12FFAR1FFAR4MAOBKEAP1
SCHEMBL8026644 0.92 NOX1 (0.52) MMP12FFAR1FFAR4MAOBKEAP1
SCHEMBL8010404 0.92 FFAR1 (0.49) MMP12FFAR1FFAR4MAOBKEAP1
SCHEMBL8026747 0.92 ALOX5 (0.52) MMP12FFAR1FFAR4MAOBALOX5
SCHEMBL8024699 0.90 FFAR1 (0.43) MMP12FFAR1FFAR4MAOB
SCHEMBL8021316 0.90 NPC1 (0.49) MMP12FFAR1FFAR4MAOBKEAP1
SCHEMBL8024571 0.89 FFAR1 (0.46) MMP12FFAR1FFAR4MAOBKEAP1
SCHEMBL8024296 0.89 NOX1 (0.48) MMP12MAOBLMNA
SCHEMBL8021221 0.89 MEN1 (0.48) MMP12FFAR1FFAR4MAOBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US claimed
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed