SCHEMBL8020340

SCHEMBL8020340

O=C(O)CN(C(=O)C(CS)CCc1ccccc1)c1ccc(OCc2ccccc2)cc1

nearest known ligand 0.71

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MMP12 P39900 1/20 0.48
FFAR1 O14842 3/20 0.48
FFAR4 Q5NUL3 1/20 0.48
KEAP1 Q14145 1/20 0.47
MAOB P27338 1/20 0.46
NOX1 Q9Y5S8 2/20 0.44
ALOX5 P09917 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8024336 0.99 FFAR1 (0.50) MMP12FFAR1FFAR4KEAP1MAOB
SCHEMBL8010235 0.96 MMP12 (0.47) MMP12FFAR1FFAR4KEAP1MAOB
SCHEMBL8026747 0.94 ALOX5 (0.52) MMP12FFAR1FFAR4MAOBALOX5
SCHEMBL8026644 0.94 NOX1 (0.52) MMP12FFAR1FFAR4KEAP1MAOB
SCHEMBL8021316 0.94 NPC1 (0.49) MMP12FFAR1FFAR4KEAP1MAOB
SCHEMBL8010404 0.94 FFAR1 (0.49) MMP12FFAR1FFAR4KEAP1MAOB
SCHEMBL8024571 0.91 FFAR1 (0.46) MMP12FFAR1FFAR4KEAP1MAOB
SCHEMBL8021221 0.91 MEN1 (0.48) MMP12FFAR1FFAR4KEAP1MAOB
SCHEMBL8024296 0.91 NOX1 (0.48) MMP12MAOBNOX1
SCHEMBL8027041 0.90 GPR132 (0.45) MMP12KEAP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US claimed
US-6156774-A Beta-thiopropionyl-amino acid derivatives and their use as beta-lactamase inhibitors SMITHKLINE BEECHAM P.L.C. (GB) 2000-12-05 US disclosed