SCHEMBL8028301

SCHEMBL8028301

COc1cc(C(F)(F)F)c(C(=O)NC(=O)N(C)C)cc1O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APP P05067 1/20 0.39
S1PR1 P21453 7/20 0.37
TMPRSS4 Q9NRS4 2/20 0.36
LMNA P02545 3/20 0.36
MAPT P10636 3/20 0.36
KDM4E B2RXH2 2/20 0.36
CYP3A4 P08684 1/20 0.36
HPGD P15428 1/20 0.36
RECQL P46063 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LRRK2 Q5S007 3/20 0.36
GAA P10253 3/20 0.34
ADRB2 P07550 1/20 0.34
GPR183 P32249 1/20 0.34
APLNR P35414 1/20 0.34
S1PR5 Q9H228 1/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8037833 0.87 SMO (0.39) APPS1PR1TMPRSS4LMNAMAPT
SCHEMBL8038215 0.86 S1PR1 (0.40) APPS1PR1TMPRSS4LMNAMAPT
SCHEMBL8041698 0.86 CYP1A2 (0.41) APPS1PR1TMPRSS4LMNAMAPT
SCHEMBL8041701 0.86 APP (0.38) APPS1PR1LMNAMAPTLRRK2
SCHEMBL8037366 0.85 S1PR1 (0.41) APPS1PR1LMNAMAPTKDM4E
SCHEMBL8033842 0.84 RAB9A (0.42) S1PR1MAPTCYP3A4HPGDMEN1
SCHEMBL8035717 0.82 ALDH1A1 (0.45) S1PR1LMNAMAPTKDM4ECYP3A4
SCHEMBL8037447 0.81 S1PR1 (0.41) APPS1PR1TMPRSS4MAPTKDM4E
SCHEMBL8037438 0.80 S1PR1 (0.45) APPS1PR1LMNAKDM4EGAA
SCHEMBL8037239 0.79 CFTR (0.47) APPTMPRSS4LMNAMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed