SCHEMBL8041701

SCHEMBL8041701

CCCN(C)C(=O)NC(=O)c1cc(O)c(OC)cc1C(F)(F)F

nearest known ligand 0.38

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
APP P05067 6/20 0.38
LRRK2 Q5S007 4/20 0.35
S1PR1 P21453 3/20 0.35
GAA P10253 1/20 0.35
LMNA P02545 1/20 0.34
RBP4 P02753 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
THRA P10827 1/20 0.33
THRB P10828 1/20 0.33
MAPT P10636 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028301 0.86 APP (0.39) APPLRRK2S1PR1GAALMNA
SCHEMBL8041698 0.85 CYP1A2 (0.41) APPLRRK2S1PR1GAALMNA
SCHEMBL8035717 0.83 ALDH1A1 (0.45) S1PR1GAALMNAMAPT
SCHEMBL8035586 0.81 SMPD1 (0.45) APPRBP4
SCHEMBL8037833 0.81 SMO (0.39) APPLRRK2S1PR1LMNAMAPT
SCHEMBL8038215 0.80 S1PR1 (0.40) APPLRRK2S1PR1GAALMNA
SCHEMBL8037415 0.79 S1PR1 (0.41) APPS1PR1GAA
SCHEMBL8037366 0.79 S1PR1 (0.41) APPS1PR1GAALMNAMAPT
SCHEMBL8033842 0.78 RAB9A (0.42) S1PR1MAPT
SCHEMBL8037435 0.77 PDE10A (0.41) APPS1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed