SCHEMBL8037833

SCHEMBL8037833

COc1cc(C(F)(F)F)c(C(=O)NC(=O)N(C)C2CC2)cc1O

nearest known ligand 0.39

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SMO Q99835 2/20 0.39
APP P05067 1/20 0.36
POLB P06746 1/20 0.34
RAB9A P51151 1/20 0.34
S1PR1 P21453 4/20 0.34
PDE4D Q08499 1/20 0.34
LRRK2 Q5S007 3/20 0.33
TMPRSS4 Q9NRS4 1/20 0.33
CCR2 P41597 1/20 0.33
CNR2 P34972 1/20 0.33
EPHX2 P34913 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 1/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
RECQL P46063 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PYGL P06737 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033842 0.94 RAB9A (0.42) SMOPOLBRAB9AS1PR1PDE4D
SCHEMBL8028301 0.87 APP (0.39) APPRAB9AS1PR1LRRK2TMPRSS4
SCHEMBL8038215 0.83 S1PR1 (0.40) APPRAB9AS1PR1LRRK2TMPRSS4
SCHEMBL8041698 0.81 CYP1A2 (0.41) APPS1PR1LRRK2TMPRSS4KDM4E
SCHEMBL8041701 0.81 APP (0.38) APPS1PR1LRRK2LMNAMAPT
SCHEMBL8040252 0.80 ALDH1A1 (0.41) POLBS1PR1LRRK2KDM4ELMNA
SCHEMBL8035618 0.80 APP (0.44) SMOAPPRAB9AKDM4EHPGD
SCHEMBL8040276 0.80 SMO (0.34) SMOAPPPOLBRAB9APDE4D
SCHEMBL8037366 0.80 S1PR1 (0.41) APPS1PR1KDM4ELMNACYP3A4
SCHEMBL8037831 0.77 ALDH1A1 (0.48) POLBRAB9ALMNAMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed