SCHEMBL8028400

SCHEMBL8028400

CC(C)(C)c1cc(-c2cc(C(C)(C)C)cc(C(C)(C)C)c2OC(P)(c2ccccc2)c2ccccc2)c(OC(P)(c2ccccc2)c2ccccc2)c(C(C)(C)C)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
TSHR P16473 1/20 0.35
CYP2C19 P33261 1/20 0.35
RXRA P19793 7/20 0.34
RXRB P28702 5/20 0.34
RXRG P48443 5/20 0.34
ALDH1A1 P00352 2/20 0.33
NPC1 O15118 1/20 0.33
PLA2G1B P04054 1/20 0.33
NFKB1 P19838 1/20 0.33
CASP3 P42574 1/20 0.33
RAB9A P51151 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SENP8 Q96LD8 1/20 0.33
SENP7 Q9BQF6 1/20 0.33
SENP6 Q9GZR1 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12355667 0.76 HSP90AA1 (0.38) CYP1A2RXRARXRBRXRGALDH1A1
SCHEMBL14586980 0.71 CYP1A2 (0.35) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL14817161 0.70 RARG (0.40) CYP3A4TSHRRXRAALDH1A1HSP90AA1
SCHEMBL30503395 0.70 CYP1A2 (0.36) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL6899796 0.70 CYP1A2 (0.35) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL11525106 0.70 CYP1A2 (0.37) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL8028404 0.69 RXRA (0.38) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL13626997 0.67 LMNA (0.33) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL8026520 0.67 MEN1 (0.47) CYP1A2CYP3A4CYP2C9TSHRCYP2C19
SCHEMBL23143159 0.67 RXRA (0.50) CYP3A4RXRARXRBRXRGRARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0653431-B1 Bis-(phosphinoalkoxy)-biaryl compounds and a process for preparing them CELANESE CHEM EUROPE GMBH (DE) 2000-03-01 EP disclosed
US-5498797-A Bis(phosphinozlkoxy)biaryl compounds and a process for their preparation HOECHST AKTIENGESELLSCHAFT (DE) 1996-03-12 US disclosed
EP-0653431-A1 Bis-(phosphinoalkoxy)-biaryl compounds and a process for preparing them HOECHST AKTIENGESELLSCHAFT (DE) 1995-05-17 EP disclosed