SCHEMBL8029642

SCHEMBL8029642

CCCC(CN1CCN(Cc2ccccc2)CC1)Oc1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 5/20 0.54
ALDH1A1 P00352 2/20 0.48
DRD4 P21917 1/20 0.48
CACNA1G O43497 2/20 0.47
KCNH2 Q12809 2/20 0.47
KDM4E B2RXH2 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
NPC1 O15118 2/20 0.46
TP53 P04637 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
LMNA P02545 1/20 0.43
MAPK1 P28482 1/20 0.43
MC4R P32245 1/20 0.43
RAB9A P51151 1/20 0.43
BCHE P06276 1/20 0.43
ACHE P22303 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029639 0.92 SIGMAR1 (0.50) SIGMAR1ALDH1A1DRD4KDM4EMEN1
SCHEMBL8029908 0.87 SIGMAR1 (0.53) SIGMAR1ALDH1A1CACNA1GKDM4EMEN1
SCHEMBL8033363 0.85 HRH3 (0.49) SIGMAR1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL8031421 0.85 SIGMAR1 (0.48) SIGMAR1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL8035801 0.82 NPC1 (0.46) SIGMAR1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL8029935 0.82 SIGMAR1 (0.59) SIGMAR1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL8035719 0.82 LTA4H (0.63) SIGMAR1ALDH1A1DRD4CACNA1GKCNH2
SCHEMBL8031455 0.81 SIGMAR1 (0.53) SIGMAR1ALDH1A1DRD4KDM4EMEN1
SCHEMBL8029877 0.80 SIGMAR1 (0.50) SIGMAR1ALDH1A1CACNA1GKCNH2KDM4E
SCHEMBL8020085 0.80 LMNA (0.59) SIGMAR1ALDH1A1KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0702010-B1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-03-15 EP disclosed
US-5668138-A AFFINITY FOR SIGMA RECEPTORS, CENTRAL NERVOUS SYSTEM DISORDERS ADIR ET COMPAGNIE (FR) 1997-09-16 US disclosed
EP-0702010-A1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-03-20 EP disclosed