SCHEMBL8034167

SCHEMBL8034167

COc1cc(Cl)c(C(=O)N(C)C(=O)N2CCCCC2)cc1OCc1ccccc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
APP P05067 7/20 0.51
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
SCN9A Q15858 2/20 0.46
HPGD P15428 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
SRD5A1 P18405 1/20 0.42
SRD5A2 P31213 1/20 0.42
RAF1 P04049 1/20 0.42
MAP2K1 Q02750 1/20 0.42
TLR9 Q9NR96 1/20 0.42
TLR7 Q9NYK1 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8031648 0.90 SMN1; SMN2 (0.52) APPNPC1RAB9AMEN1KMT2A
SCHEMBL8038345 0.82 HPGD (0.52) APPNPC1RAB9AMEN1KMT2A
SCHEMBL8031650 0.81 MEN1 (0.46) APPNPC1RAB9AMEN1KMT2A
SCHEMBL8034163 0.81 CTSV (0.47) APPNPC1RAB9AMEN1KMT2A
SCHEMBL8022341 0.81 MEN1 (0.50) APPNPC1RAB9AMEN1KMT2A
SCHEMBL8022338 0.79 TRPM8 (0.46) APPNPC1RAB9AMEN1KMT2A
SCHEMBL8035938 0.79 SRD5A1 (0.47) APPNPC1RAB9AMEN1KMT2A
SCHEMBL8034161 0.79 APP (0.47) APPNPC1RAB9AMEN1KMT2A
SCHEMBL8039013 0.79 ALDH1A1 (0.41) RAB9AMEN1KMT2AHPGDSMN1; SMN2
SCHEMBL8037071 0.78 MEN1 (0.47) APPNPC1RAB9AMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed