SCHEMBL8034979

SCHEMBL8034979

COCCCN(C(=O)NC1CC1)C(=O)c1cc(OCc2ccccc2)c(OC)cc1C(F)(F)F

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 2/20 0.40
SGMS2 Q8NHU3 1/20 0.39
NPC1 O15118 2/20 0.39
PKM P14618 1/20 0.39
RAB9A P51151 1/20 0.39
LMNA P02545 1/20 0.38
SMPD1 P17405 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC8 Q9BY41 1/20 0.38
HDAC6 Q9UBN7 1/20 0.38
BRD4 O60885 1/20 0.38
REN P00797 3/20 0.37
TRPM8 Q7Z2W7 3/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
PTK2 Q05397 1/20 0.36
CYP3A4 P08684 1/20 0.36
CTSV O60911 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8032754 0.95 MEN1 (0.41) MEN1KMT2AALDH1A1SGMS2NPC1
SCHEMBL8039272 0.91 TRPM8 (0.41) MEN1KMT2AALDH1A1SGMS2NPC1
SCHEMBL8031645 0.89 NPC1 (0.41) MEN1KMT2AALDH1A1SGMS2NPC1
SCHEMBL8039269 0.85 ALDH1A1 (0.43) MEN1KMT2AALDH1A1SGMS2NPC1
SCHEMBL8035584 0.83 LRRK2 (0.36) ALDH1A1APPPDE4B
SCHEMBL8025483 0.80 MEN1 (0.46) MEN1KMT2AALDH1A1SGMS2NPC1
SCHEMBL8034971 0.79 MTNR1B (0.44) MEN1KMT2AALDH1A1NPC1LMNA
SCHEMBL8031681 0.78 LRRK2 (0.38) ALDH1A1APPPDE4B
SCHEMBL8039007 0.77 PTGES (0.41) ALDH1A1PKMLMNACYP3A4
SCHEMBL8035618 0.77 APP (0.44) MEN1KMT2ANPC1PKMRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed