SCHEMBL8041806

SCHEMBL8041806

O=C(O)Cn1nnnc1Sc1ncc(C(=O)O)s1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
RXRA P19793 1/20 0.38
RXRB P28702 1/20 0.38
RXRG P48443 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
ALDH1A1 P00352 3/20 0.36
HPGD P15428 1/20 0.36
MAPK1 P28482 2/20 0.36
GLA P06280 1/20 0.36
MAPT P10636 1/20 0.36
HCAR2 Q8TDS4 1/20 0.36
USP7 Q93009 1/20 0.33
POLB P06746 1/20 0.32
LMNA P02545 2/20 0.31
KDM4E B2RXH2 1/20 0.31
MEN1 O00255 1/20 0.31
HSD17B10 Q99714 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
TSHR P16473 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8042980 0.87 ALDH1A1 (0.41) KMT2ANPC1RXRARXRBRXRG
SCHEMBL8042788 0.85 HSD17B10 (0.42) KMT2ANPC1RXRARXRBRXRG
SCHEMBL8051020 0.85 KDM4C (0.38) KMT2ANPC1KDM4CALDH1A1HPGD
SCHEMBL8033764 0.83 HTT (0.46) KMT2ARXRARXRBRXRGALDH1A1
SCHEMBL8046221 0.83 ALDH1A1 (0.51) KMT2AALDH1A1HPGDMAPK1MAPT
SCHEMBL8050401 0.81 KMT2A (0.36) KMT2ANPC1KDM4CALDH1A1HPGD
SCHEMBL8050397 0.81 ALDH1A1 (0.40) KMT2ARXRARXRBRXRGKDM4C
SCHEMBL8032474 0.81 NPC1 (0.47) KMT2ANPC1KDM4CALDH1A1HPGD
SCHEMBL8043875 0.80 UBE2M (0.37) RXRARXRBRXRGALDH1A1HPGD
SCHEMBL8716288 0.80 CYP2C19 (0.47) KMT2ARXRARXRBRXRGALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed