SCHEMBL8043221

SCHEMBL8043221

Cc1ccc(S(=O)(=O)Cc2nnc(Sc3nc4ccc([N+](=O)[O-])cc4s3)n2-c2ccccc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 1/20 0.44
MAPT P10636 8/20 0.42
HTT P42858 6/20 0.42
SMN1; SMN2 Q16637 4/20 0.42
ALDH1A1 P00352 4/20 0.42
KMT2A Q03164 3/20 0.42
MEN1 O00255 1/20 0.42
LMNA P02545 2/20 0.42
MAPK1 P28482 2/20 0.42
CA2 P00918 2/20 0.42
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
NPSR1 Q6W5P4 3/20 0.41
CYP3A4 P08684 2/20 0.40
CYP1A2 P05177 1/20 0.40
TSHR P16473 1/20 0.40
TP53 P04637 1/20 0.40
KEAP1 Q14145 1/20 0.40
TDP1 Q9NUW8 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033626 0.88 KMT2A (0.42) MAPTHTTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL8043682 0.88 HTT (0.50) MAPTHTTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL8047470 0.86 ALDH1A1 (0.40) MAPTHTTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL8715778 0.80 HTT (0.42) MAPTHTTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL8046037 0.79 NPC1 (0.42) MAPTHTTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL8044246 0.78 ALDH1A1 (0.39) MAPTHTTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL8041911 0.78 PDK1 (0.51) PDK1MAPTHTTSMN1; SMN2ALDH1A1
SCHEMBL8042500 0.78 KDM4E (0.38) MAPTHTTSMN1; SMN2ALDH1A1KMT2A
SCHEMBL8048212 0.78 PDK1 (0.48) PDK1MAPTHTTSMN1; SMN2ALDH1A1
SCHEMBL8034272 0.77 ALDH1A1 (0.41) MAPTHTTSMN1; SMN2ALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed