SCHEMBL8046037

SCHEMBL8046037

Cc1ccc(S(=O)(=O)Cc2nnc(Sc3ncc([N+](=O)[O-])s3)n2-c2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.42
RAB9A P51151 3/20 0.42
TLR9 Q9NR96 3/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
AGTR1 P30556 2/20 0.42
KEAP1 Q14145 2/20 0.41
ALDH1A1 P00352 6/20 0.39
MAPK8 P45983 6/20 0.38
MAPK9 P45984 6/20 0.38
SIRT2 Q8IXJ6 2/20 0.38
MAPK10 P53779 2/20 0.38
HTT P42858 3/20 0.37
NPSR1 Q6W5P4 3/20 0.37
S1PR4 O95977 2/20 0.37
MAPT P10636 2/20 0.37
S1PR1 P21453 2/20 0.37
MAPK1 P28482 2/20 0.37
TDP1 Q9NUW8 1/20 0.37
HSP90AA1 P07900 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044438 0.86 ALDH1A1 (0.41) KMT2AKEAP1ALDH1A1HTTNPSR1
SCHEMBL8052232 0.85 ALDH1A1 (0.43) MEN1KMT2AKEAP1ALDH1A1HTT
SCHEMBL8046773 0.84 PKM (0.41) MEN1KMT2AALDH1A1HTTNPSR1
SCHEMBL8043961 0.80 ALDH1A1 (0.42) MEN1KMT2AALDH1A1HTTNPSR1
SCHEMBL8050394 0.80 ALDH1A1 (0.41) MEN1KMT2AALDH1A1HTTNPSR1
SCHEMBL8043221 0.79 PDK1 (0.44) NPC1MEN1KMT2AKEAP1ALDH1A1
SCHEMBL8043682 0.79 HTT (0.50) NPC1RAB9AKMT2AALDH1A1HTT
SCHEMBL8034272 0.79 ALDH1A1 (0.41) NPC1RAB9AMEN1KMT2AALDH1A1
SCHEMBL8044246 0.79 ALDH1A1 (0.39) KMT2AALDH1A1HTTNPSR1MAPT
SCHEMBL8032480 0.76 PKM (0.38) MEN1KMT2AALDH1A1HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed