SCHEMBL8043493

SCHEMBL8043493

CCc1nc(-c2ccc(Cl)cc2)nc(NC2CCCCC2)c1C(=O)O

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
PLA2G1B P04054 1/20 0.45
ATG4B Q9Y4P1 1/20 0.45
RXRA P19793 1/20 0.43
NR4A2 P43354 1/20 0.43
PDE5A O76074 2/20 0.43
ACP1 P24666 2/20 0.43
CNR1 P21554 5/20 0.40
FABP3 P05413 1/20 0.39
FABP4 P15090 1/20 0.39
FABP5 Q01469 1/20 0.39
ADORA3 P0DMS8 2/20 0.39
ADORA1 P30542 2/20 0.39
ADORA2A P29274 1/20 0.39
KDM4E B2RXH2 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
POLB P06746 2/20 0.39
CNR2 P34972 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8034844 0.88 CASP3 (0.46) PLA2G1BATG4BRXRANR4A2ADORA3
SCHEMBL8037126 0.87 PLA2G1B (0.41) PLA2G1BATG4BRXRANR4A2PDE5A
SCHEMBL8030010 0.81 RXRA (0.47) RXRANR4A2ACP1FABP3FABP4
SCHEMBL4011568 0.80 FABP4 (0.42) RXRANR4A2FABP3FABP4FABP5
SCHEMBL8038516 0.77 NPSR1 (0.39) PLA2G1BATG4BPDE5AACP1CNR1
SCHEMBL8040520 0.76 NPSR1 (0.43) PLA2G1BATG4BRXRANR4A2ACP1
SCHEMBL5961069 0.76 FABP3 (0.49) RXRANR4A2FABP3FABP4FABP5
SCHEMBL8037000 0.76 RXRA (0.47) RXRANR4A2FABP3FABP4FABP5
SCHEMBL4151850 0.74 FABP3 (0.48) RXRANR4A2ACP1FABP3FABP4
SCHEMBL14914473 0.74 PPARG (0.54) ADORA1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009080242-A1 SUBSTITUTED 4-AMINOPYRIMIDINE-5-CARBOXYLIC ACID AND USE THEREOF BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2009-07-02 WO disclosed