SCHEMBL8043580

SCHEMBL8043580

CCCCn1nnnc1Sc1nc(C(F)(F)F)c(C(=O)O)s1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.43
CYP2C19 P33261 2/20 0.42
KMT2A Q03164 4/20 0.41
MEN1 O00255 3/20 0.41
ALDH1A1 P00352 10/20 0.40
GAA P10253 3/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
MAPT P10636 3/20 0.39
USP2 O75604 2/20 0.39
LMNA P02545 2/20 0.39
TSHR P16473 2/20 0.39
ATM Q13315 1/20 0.39
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
PKM P14618 1/20 0.37
NPSR1 Q6W5P4 1/20 0.34
HSD17B10 Q99714 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033927 0.93 NPSR1 (0.40) HTTCYP2C19KMT2AMEN1ALDH1A1
SCHEMBL8033964 0.89 SMN1; SMN2 (0.39) HTTCYP2C19KMT2AMEN1ALDH1A1
SCHEMBL8043236 0.89 UBE2M (0.35) HTTALDH1A1
SCHEMBL8034114 0.86 HTT (0.31) HTTCYP2C19ALDH1A1
SCHEMBL8033786 0.84 MAPT (0.39) KMT2AALDH1A1HPGDMAPTLMNA
SCHEMBL8051249 0.84 RAB9A (0.35) HTTALDH1A1GAAPOLBHPGD
SCHEMBL8042294 0.82 ALDH1A1 (0.38) HTTKMT2AMEN1ALDH1A1GAA
SCHEMBL8043035 0.80 MAPT (0.33) ALDH1A1POLBMAPTLMNA
SCHEMBL8042982 0.80 KMT2A (0.35) HTTCYP2C19KMT2AMEN1ALDH1A1
SCHEMBL8042593 0.80 ALDH1A1 (0.47) HTTKMT2AMEN1ALDH1A1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed