SCHEMBL8043817

SCHEMBL8043817

CCc1nnc(Sc2ncc(S(C)(=O)=O)s2)s1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 5/20 0.37
MAPK9 P45984 5/20 0.37
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
LOXL2 Q9Y4K0 8/20 0.35
NPC1 O15118 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
CA4 P22748 1/20 0.35
CA5A P35218 1/20 0.35
CA5B Q9Y2D0 1/20 0.35
ATM Q13315 1/20 0.33
MAPK10 P53779 1/20 0.33
KDM4E B2RXH2 1/20 0.33
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
KMT2A Q03164 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
LOX P28300 1/20 0.33
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8048119 0.89 MAPK8 (0.38) MAPK8MAPK9LOXL2MAPK10ALDH1A1
SCHEMBL8041884 0.88 MAPK8 (0.36) MAPK8MAPK9LOXL2NPC1MAPK10
SCHEMBL8042354 0.87 MAPK8 (0.34) MAPK8MAPK9LOXL2MAPK10LOX
SCHEMBL8044752 0.85 MAPK8 (0.33) MAPK8MAPK9LOXL2MAPK10LOX
SCHEMBL8044039 0.85 ALDH1A1 (0.37) MAPK8MAPK9LOXL2MAPK10MEN1
SCHEMBL8043583 0.84 AKT1 (0.33) MAPK8MAPK9LOXL2MAPK10LOX
SCHEMBL8043647 0.83 F2 (0.40) MAPK8MAPK9LOXL2MAPK10ALDH1A1
SCHEMBL8043608 0.82 APEX1 (0.33) MAPK8MAPK9ALDH1A1
SCHEMBL8044491 0.82 LMNA (0.48) MAPTLOXL2NPC1MEN1ALDH1A1
SCHEMBL8042764 0.81 SMN1; SMN2 (0.42) MAPTMEN1ALDH1A1KMT2AAKT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed