SCHEMBL8044449

SCHEMBL8044449

CCOC(=O)Cc1nnc(Sc2ncc(C(=O)O)s2)s1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.43
HSD17B10 Q99714 3/20 0.43
USP2 O75604 2/20 0.43
POLB P06746 4/20 0.42
RXRA P19793 1/20 0.41
RXRB P28702 1/20 0.41
RXRG P48443 1/20 0.41
RECQL P46063 1/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
MAPT P10636 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
HCAR2 Q8TDS4 1/20 0.39
HTT P42858 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8044854 0.88 RXRA (0.39) SMN1; SMN2HSD17B10USP2POLBRXRA
SCHEMBL8042807 0.84 MEN1 (0.44) SMN1; SMN2HSD17B10USP2POLBRECQL
SCHEMBL8042939 0.83 RXRA (0.41) RXRARXRBRXRGHCAR2GAA
SCHEMBL8050209 0.83 RXRA (0.43) HSD17B10POLBRXRARXRBRXRG
SCHEMBL8042764 0.81 SMN1; SMN2 (0.42) SMN1; SMN2HSD17B10USP2POLBRECQL
SCHEMBL8044684 0.81 RXRA (0.42) POLBRXRARXRBRXRGRECQL
SCHEMBL8043440 0.81 F2 (0.43) RXRARXRBRXRGALDH1A1HCAR2
SCHEMBL8033917 0.81 MAPK8 (0.56) SMN1; SMN2HSD17B10USP2POLBMEN1
SCHEMBL8044327 0.80 RXRA (0.41) SMN1; SMN2HSD17B10POLBRXRARXRB
SCHEMBL8046385 0.80 RXRA (0.41) RXRARXRBRXRGMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed