SCHEMBL8048034

SCHEMBL8048034

CC(C)(C)c1cccc(C2=NC(=S)N=N2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.49
RXRA P19793 2/20 0.41
RXRB P28702 2/20 0.41
OPRD1 P41143 3/20 0.35
CTSS P25774 1/20 0.35
CTSK P43235 1/20 0.35
OPRM1 P35372 1/20 0.35
OPRK1 P41145 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
TMEM97 Q5BJF2 1/20 0.34
SIGMAR1 Q99720 1/20 0.34
MPL P40238 1/20 0.33
PTAFR P25105 1/20 0.33
ABCG2 Q9UNQ0 1/20 0.33
ACHE P22303 3/20 0.33
CTSA P10619 1/20 0.32
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8041917 0.83 CTSS (0.44) CTSS
SCHEMBL8047010 0.79 KIF11 (0.44) KIF11
SCHEMBL8042855 0.74 ALDH1A1 (0.45)
SCHEMBL8047366 0.74 TAAR1 (0.40) CYP3A4
SCHEMBL5547288 0.73 KIF11 (0.72) KIF11RXRARXRBOPRD1CTSS
SCHEMBL30023786 0.73 KIF11 (0.72) KIF11RXRARXRBOPRD1CTSS
SCHEMBL27659191 0.71 KIF11 (0.76) KIF11RXRARXRBOPRD1CTSS
SCHEMBL25666511 0.70 KIF11 (0.49) KIF11RXRARXRBOPRD1CTSS
SCHEMBL25706667 0.69 KIF11 (0.67) KIF11RXRARXRBOPRD1CTSS
SCHEMBL25616851 0.68 KIF11 (0.55) KIF11RXRARXRBOPRD1CTSS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed