SCHEMBL8052167

SCHEMBL8052167

Cc1cc(-n2nnnc2Sc2nc3ccc(C(=O)O)cc3s2)sc1C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.41
HTT P42858 3/20 0.41
MEN1 O00255 7/20 0.40
KMT2A Q03164 7/20 0.40
MAPT P10636 6/20 0.40
HPGD P15428 7/20 0.40
SMN1; SMN2 Q16637 4/20 0.39
NFKB1 P19838 3/20 0.39
NFKB2 Q00653 3/20 0.39
RELA Q04206 3/20 0.39
KDM4E B2RXH2 2/20 0.39
LMNA P02545 2/20 0.39
NPC1 O15118 3/20 0.38
RAB9A P51151 3/20 0.38
MITF O75030 2/20 0.38
TP53 P04637 2/20 0.38
PTPN1 P18031 1/20 0.38
ILK Q13418 1/20 0.37
POLB P06746 3/20 0.37
RECQL P46063 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8047829 0.87 ALDH1A1 (0.40) ALDH1A1HTTMEN1KMT2AMAPT
SCHEMBL8033820 0.83 ALDH1A1 (0.49) ALDH1A1HTTMEN1KMT2AMAPT
SCHEMBL8042685 0.83 NFKB1 (0.42) ALDH1A1HTTMEN1KMT2AMAPT
SCHEMBL8046550 0.83 ALDH1A1 (0.40) ALDH1A1HTTMEN1KMT2AMAPT
SCHEMBL8044411 0.83 KMT2A (0.55) ALDH1A1HTTMEN1KMT2AMAPT
SCHEMBL8033619 0.82 PKM (0.40) ALDH1A1HTTMEN1KMT2AMAPT
SCHEMBL8033225 0.82 ALDH1A1 (0.47) ALDH1A1HTTMEN1KMT2AMAPT
SCHEMBL8042977 0.82 PDK1 (0.51) ALDH1A1HTTMEN1KMT2AMAPT
SCHEMBL8042101 0.81 HPGD (0.45) ALDH1A1MEN1KMT2AMAPTHPGD
SCHEMBL8043375 0.81 SMN1; SMN2 (0.45) ALDH1A1MEN1KMT2AMAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed