SCHEMBL8046550

SCHEMBL8046550

O=C(O)c1ccc2nc(Sc3nnnn3-c3ccc(Br)s3)sc2c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 8/20 0.40
HPGD P15428 7/20 0.40
MEN1 O00255 7/20 0.40
KMT2A Q03164 7/20 0.40
NFKB1 P19838 3/20 0.40
NFKB2 Q00653 3/20 0.40
RELA Q04206 3/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
KDM4E B2RXH2 2/20 0.40
LMNA P02545 2/20 0.40
MAPT P10636 5/20 0.38
POLB P06746 2/20 0.38
NPC1 O15118 2/20 0.38
MITF O75030 2/20 0.38
RAB9A P51151 2/20 0.38
RECQL P46063 2/20 0.38
GAA P10253 1/20 0.38
GFER P55789 1/20 0.38
PAX8 Q06710 1/20 0.38
KLF5 Q13887 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8047829 0.88 ALDH1A1 (0.40) ALDH1A1HPGDMEN1KMT2ANFKB1
SCHEMBL8048432 0.85 MEN1 (0.47) ALDH1A1HPGDMEN1KMT2ANFKB1
SCHEMBL8044245 0.85 MEN1 (0.46) ALDH1A1HPGDMEN1KMT2ANFKB1
SCHEMBL8033820 0.84 ALDH1A1 (0.49) ALDH1A1HPGDMEN1KMT2ANFKB1
SCHEMBL8042685 0.84 NFKB1 (0.42) ALDH1A1HPGDMEN1KMT2ANFKB1
SCHEMBL8044411 0.83 KMT2A (0.55) ALDH1A1HPGDMEN1KMT2ANFKB1
SCHEMBL8052167 0.83 ALDH1A1 (0.41) ALDH1A1HPGDMEN1KMT2ANFKB1
SCHEMBL8047942 0.81 PKM (0.40) ALDH1A1HPGDMEN1KMT2ASMN1; SMN2
SCHEMBL8043758 0.81 PDK1 (0.52) ALDH1A1MEN1KMT2ASMN1; SMN2LMNA
SCHEMBL8044849 0.81 ALDH1A1 (0.49) ALDH1A1HPGDKMT2ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed