SCHEMBL8059176

SCHEMBL8059176

CP(=O)(O)C(Cc1ccsc1)(C(=O)O)c1ccccc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 2/20 0.38
OPRD1 P41143 2/20 0.38
OPRK1 P41145 2/20 0.38
GRM5 P41594 1/20 0.37
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
GRM2 Q14416 1/20 0.34
GRM3 Q14832 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HIF1A Q16665 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A3 Q01959 1/20 0.34
POLB P06746 1/20 0.34
CHRM2 P08172 1/20 0.34
CHRM1 P11229 1/20 0.34
CHRM3 P20309 1/20 0.34
TDP1 Q9NUW8 1/20 0.33
HPGD P15428 1/20 0.33
FDPS P14324 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8046595 0.87 OPRM1 (0.36) OPRM1OPRD1OPRK1GRM5L3MBTL1
SCHEMBL8059146 0.85 CETP (0.36) OPRM1OPRD1OPRK1GRM5L3MBTL1
SCHEMBL8058487 0.78 FDPS (0.46) SMN1; SMN2POLBFDPSMAPT
SCHEMBL8058488 0.77 HPGD (0.41) SMN1; SMN2POLBTDP1HPGDCYP1A2
SCHEMBL8059117 0.75 FDPS (0.58) HIF1AFDPSMAPTCYP1A2CYP2C9
SCHEMBL7746842 0.72 OPRM1 (0.42) OPRM1OPRD1OPRK1GRM5L3MBTL1
SCHEMBL8059181 0.71 FDPS (0.52) SMN1; SMN2POLBFDPSCYP1A2CYP2C19
SCHEMBL8059151 0.70 GRM2 (0.38) OPRM1OPRD1OPRK1GRM5GRM2
SCHEMBL10806221 0.70 OPRM1 (0.42) OPRM1OPRD1OPRK1HDAC8HDAC6
SCHEMBL27788552 0.70 OPRM1 (0.42) OPRM1OPRD1OPRK1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6046180-A NAALADase inhibitors GUILFORD PHARMACEUTICALS INC. (US) 2000-04-04 US disclosed
EP-0936914-A1 HYDROXY-PHOSPHINYL DERIVATIVES USEFUL AS NAALADASE INHIBITORS GUILFORD PHARMACEUTICALS INC. (US) 1999-08-25 EP disclosed
EP-0936914-A4 1999-08-25 EP disclosed
WO-1997048400-A1 HYDROXY-PHOSPHINYL DERIVATIVES USEFUL AS NAALADASE INHIBITORS GUILFORD PHARMACEUTICALS INC. (US) 1997-12-24 WO disclosed