SCHEMBL8062877

SCHEMBL8062877

O=C(NCC1CCN(S(=O)(=O)c2ccc(-c3ccccc3)cc2)CC1)N[C@@]12C[C@@H]3C[C@@H]4C[C@H](C1)C2(C4)C3

nearest known ligand 0.50

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.50
L3MBTL1 Q9Y468 1/20 0.50
EPHX1 P07099 9/20 0.46
EPHX2 P34913 9/20 0.46
KDM1A O60341 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
PKM P14618 1/20 0.41
POLB P06746 1/20 0.39
USP5 P45974 1/20 0.39
HTR2B P41595 1/20 0.39
TGM2 P21980 2/20 0.39
F13A1 P00488 1/20 0.39
TGM1 P22735 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4537354 0.85 EPHX1 (0.63) ALDH1A1L3MBTL1EPHX1EPHX2
SCHEMBL4535452 0.80 EPHX2 (0.58) ALDH1A1L3MBTL1EPHX1EPHX2
SCHEMBL8064838 0.79 EPHX1 (0.68) ALDH1A1L3MBTL1EPHX1EPHX2
SCHEMBL8053617 0.79 RAB9A (0.44) EPHX1EPHX2
SCHEMBL8063484 0.79 EPHX2 (0.52) EPHX1EPHX2HDAC6
SCHEMBL8066757 0.77 ALDH1A1 (0.43) ALDH1A1L3MBTL1EPHX1EPHX2
SCHEMBL8069507 0.77 MMP2 (0.46)
SCHEMBL8061524 0.76 EPHX2 (0.49) EPHX1EPHX2HDAC6
SCHEMBL8066636 0.74 RAB9A (0.46) ALDH1A1
SCHEMBL8068354 0.74 PSEN1 (0.47) ALDH1A1L3MBTL1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009070497-A1 SEH AND 11 β-HSD1 INHIBITORS AND THEIR USE SMITHKLINE BEECHAM CORPORATION (US) 2009-06-04 WO disclosed