SCHEMBL8068481

SCHEMBL8068481

COC(=O)c1ccc(Oc2ccc(CCN(C)C)cc2)c(S(C)(=O)=O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.43
THRB P10828 1/20 0.43
POLB P06746 1/20 0.42
PKM P14618 1/20 0.42
BMP1 P13497 3/20 0.41
VCAM1 P19320 1/20 0.41
ALDH1A1 P00352 2/20 0.41
HPGD P15428 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
KMT2A Q03164 1/20 0.40
USP2 O75604 1/20 0.40
CYP1A2 P05177 1/20 0.40
TSHR P16473 1/20 0.40
CYP2C19 P33261 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
RAB9A P51151 1/20 0.40
LPAR1 Q92633 1/20 0.39
LPAR5 Q9H1C0 1/20 0.39
HRH3 Q9Y5N1 2/20 0.39
DRD2 P14416 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8068832 0.90 PKM (0.43) POLBPKMBMP1ALDH1A1HPGD
SCHEMBL8075422 0.89 PKM (0.48) THRATHRBPOLBPKMKMT2A
Hydrochloric Acid SCHEMBL8070153 0.88 PKM (0.47) THRATHRBPOLBPKMKMT2A
SCHEMBL8068841 0.86 THRA (0.40) THRATHRBPOLBPKMVCAM1
SCHEMBL8073466 0.85 BMP1 (0.40) THRATHRBBMP1LPAR1LPAR5
SCHEMBL8071065 0.84 THRA (0.44) THRATHRBPOLBPKMVCAM1
SCHEMBL8072805 0.83 SMN1; SMN2 (0.51) ALDH1A1HPGDKMT2ATSHRSMN1; SMN2
SCHEMBL8059397 0.83 THRA (0.42) THRATHRBPOLBPKMBMP1
SCHEMBL8059406 0.83 SLC9A1 (0.47)
SCHEMBL8059495 0.83 THRA (0.41) THRATHRBPOLBPKMBMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed