SCHEMBL8071065

SCHEMBL8071065

COC(=O)c1ccc(Oc2ccc(SCCN(C)C)cc2)c(S(C)(=O)=O)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
POLB P06746 1/20 0.40
PKM P14618 1/20 0.40
ALDH1A1 P00352 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
VCAM1 P19320 1/20 0.39
SLC6A4 P31645 4/20 0.39
MAPT P10636 2/20 0.39
USP2 O75604 1/20 0.38
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
RAB9A P51151 1/20 0.38
L3MBTL1 Q9Y468 2/20 0.37
CYP2C9 P11712 1/20 0.36
KMT2A Q03164 1/20 0.36
SLC6A2 P23975 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8059482 0.89 THRA (0.47) THRATHRBPOLBPKMSLC6A4
SCHEMBL8068841 0.86 THRA (0.40) THRATHRBPOLBPKMALDH1A1
SCHEMBL8068481 0.84 THRA (0.43) THRATHRBPOLBPKMALDH1A1
Hydrochloric Acid SCHEMBL8070615 0.84 THRA (0.41) THRATHRBPOLBPKMNPSR1
Hydrochloric Acid SCHEMBL8070618 0.83 SLC9A1 (0.44)
SCHEMBL8068454 0.81 THRA (0.44) THRATHRBALDH1A1HPGDNPSR1
SCHEMBL8375529 0.78 VCAM1 (0.48) ALDH1A1HPGDNPSR1VCAM1MAPT
SCHEMBL8379224 0.75 ALDH1A1 (0.54) PKMALDH1A1HPGDNPSR1VCAM1
SCHEMBL8444218 0.75 PKM (0.44) THRATHRBPOLBPKMALDH1A1
SCHEMBL8068832 0.74 PKM (0.43) POLBPKMALDH1A1HPGDNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed