SCHEMBL8068670

SCHEMBL8068670

COC(=O)c1ccc(Oc2ccc(CSCCN(C)C)cc2)c(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 1/20 0.43
SLC6A2 P23975 3/20 0.41
SLC6A4 P31645 3/20 0.41
MRGPRX4 Q96LA9 1/20 0.40
THRA P10827 1/20 0.40
THRB P10828 1/20 0.40
SIRT1 Q96EB6 1/20 0.40
CYP3A4 P08684 1/20 0.39
ESRRA P11474 1/20 0.39
ROCK2 O75116 1/20 0.38
LPAR1 Q92633 2/20 0.38
LPAR5 Q9H1C0 2/20 0.38
AR P10275 1/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
SCN9A Q15858 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MAPT P10636 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8068951 0.90 LPAR1 (0.46) SLC6A2SLC6A4MRGPRX4THRATHRB
SCHEMBL8068627 0.86 LPAR1 (0.48) NOTUMSLC6A2SLC6A4MRGPRX4THRA
SCHEMBL8068454 0.86 THRA (0.44) NOTUMSLC6A2SLC6A4MRGPRX4THRA
Hydrochloric Acid SCHEMBL8059587 0.85 SIRT1 (0.42) SLC6A2SLC6A4THRATHRBSIRT1
Hydrochloric Acid SCHEMBL8059590 0.84 SLC9A1 (0.41) SLC6A2SLC6A4THRATHRBCYP3A4
SCHEMBL8068841 0.82 THRA (0.40) SLC6A2SLC6A4THRATHRBCYP3A4
SCHEMBL12239037 0.80 LOXL2 (0.55) NOTUMSLC6A2SLC6A4MRGPRX4CYP3A4
SCHEMBL8075068 0.75 NOTUM (0.54) NOTUMMRGPRX4CYP3A4ESRRAALDH1A1
SCHEMBL8059726 0.75 THRA (0.47) SLC6A2SLC6A4MRGPRX4THRATHRB
SCHEMBL27195845 0.75 THRA (0.60) NOTUMMRGPRX4THRATHRBSIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed