SCHEMBL8070558

SCHEMBL8070558

CCC(NS(=O)(=O)c1ccc(Oc2ccc(C(=O)O)cc2S(C)(=O)=O)cc1)n1ccnc1

nearest known ligand 0.39

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP24A1 Q07973 3/20 0.39
GFER P55789 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
TBXA2R P21731 1/20 0.36
GAA P10253 1/20 0.35
ALDH1A1 P00352 1/20 0.35
AGTR2 P50052 1/20 0.35
CYP26A1 O43174 1/20 0.34
CYP3A4 P08684 1/20 0.34
KMT2A Q03164 1/20 0.34
WDR5 P61964 1/20 0.34
TDP1 Q9NUW8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8447165 0.78 NPSR1 (0.45) GFERNPSR1ALDH1A1TDP1
SCHEMBL8068480 0.78 CYP19A1 (0.55) ALDH1A1KMT2A
SCHEMBL8059431 0.75 CYP19A1 (0.51) KMT2ATDP1
SCHEMBL8070529 0.74 CYP19A1 (0.45) KMT2A
SCHEMBL8068476 0.74 CYP17A1 (0.45) CYP24A1CYP3A4
SCHEMBL8446010 0.73 MAPT (0.42) NPSR1ALDH1A1KMT2A
SCHEMBL8059678 0.73 NPSR1 (0.44) NPSR1ALDH1A1KMT2A
SCHEMBL8059681 0.72 TTR (0.45) GFERNPSR1GAA
SCHEMBL8068849 0.72 ALDH1A1 (0.54) GFERALDH1A1KMT2ATDP1
SCHEMBL8073502 0.72 TTR (0.51) NPSR1GAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed