SCHEMBL8068480

SCHEMBL8068480

CS(=O)(=O)c1cc(C(=O)O)ccc1Oc1ccc(S(=O)(=O)NCCCn2ccnc2)cc1

nearest known ligand 0.55

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.55
ALDH1A1 P00352 1/20 0.55
POLB P06746 2/20 0.54
TBXAS1 P24557 4/20 0.51
KMT2A Q03164 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8446065 0.88 CYP19A1 (0.50) CYP19A1ALDH1A1POLBKMT2A
Hydrochloric Acid SCHEMBL8070594 0.87 CYP19A1 (0.49) CYP19A1ALDH1A1POLBKMT2A
SCHEMBL8059431 0.81 CYP19A1 (0.51) CYP19A1TBXAS1KMT2A
SCHEMBL8070529 0.79 CYP19A1 (0.45) CYP19A1TBXAS1KMT2A
SCHEMBL8068849 0.78 ALDH1A1 (0.54) ALDH1A1POLBKMT2A
SCHEMBL8070558 0.78 CYP24A1 (0.39) ALDH1A1KMT2A
SCHEMBL8068934 0.78 SIGMAR1 (0.51) POLBKMT2A
SCHEMBL5564831 0.77 ALDH1A1 (0.74) CYP19A1ALDH1A1POLBTBXAS1KMT2A
SCHEMBL8073771 0.76 KMT2A (0.58) ALDH1A1POLBKMT2A
SCHEMBL8070495 0.76 KDM4E (0.67) ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6057322-A USEFUL IN TREATMENT OF CARDIOVASCULAR DISEASES HOECHST AKTIENGESELLSCHAFT (DE) 2000-05-02 US disclosed