SCHEMBL8073643

SCHEMBL8073643

Cc1nc(-c2ccc(C(=O)N3CCN(S(=O)(=O)c4ccc([N+](=O)[O-])cc4)CC3)cc2)no1.O=[N+]([O-])c1ccc(S(=O)(=O)Cl)cc1

nearest known ligand 0.56

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.56
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA2 P00918 1/20 0.48
CA7 P43166 1/20 0.48
CA9 Q16790 1/20 0.48
CA14 Q9ULX7 1/20 0.48
LMNA P02545 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
HTT P42858 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
FAAH O00519 2/20 0.45
KMT2A Q03164 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
MGLL Q99685 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7073993 0.96 ALDH1A1 (0.60) ALDH1A1CA12CA1CA2CA7
SCHEMBL8080659 0.86 LMNA (0.55) ALDH1A1CA12CA1CA2CA7
SCHEMBL7071746 0.86 MEN1 (0.54) ALDH1A1CA12CA1CA2CA7
SCHEMBL7074222 0.85 LMNA (0.62) ALDH1A1LMNASMN1; SMN2HTTNPSR1
SCHEMBL8075470 0.85 LMNA (0.46) ALDH1A1LMNASMN1; SMN2HTTNPSR1
SCHEMBL7069907 0.85 VCAM1 (0.52) LMNASMN1; SMN2KMT2AMGLL
SCHEMBL8072947 0.84 THRB (0.46) ALDH1A1LMNASMN1; SMN2HTTNPSR1
SCHEMBL7071582 0.84 LMNA (0.60) ALDH1A1LMNASMN1; SMN2HTTNPSR1
SCHEMBL7069936 0.84 SMN1; SMN2 (0.60) ALDH1A1LMNASMN1; SMN2KMT2A
SCHEMBL7075122 0.83 LMNA (0.65) ALDH1A1LMNASMN1; SMN2HTTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1025086-A1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GmbH (DE) 2000-08-09 EP disclosed
WO-1999016751-A1 BENZAMIDINE DERIVATIVES AS FACTOR XA INHIBITORS MERCK PATENT GMBH (DE) 1999-04-08 WO disclosed