SCHEMBL8074308

SCHEMBL8074308

[CH2]c1ccccc1S(=O)(=O)N(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
HTT P42858 2/20 0.53
SMN1; SMN2 Q16637 2/20 0.50
POLB P06746 2/20 0.49
LMNA P02545 2/20 0.40
MCL1 Q07820 1/20 0.40
ALOX5AP P20292 1/20 0.39
FEN1 P39748 1/20 0.39
PDPK1 O15530 1/20 0.38
ROCK2 O75116 1/20 0.38
FES P07332 1/20 0.38
FER P16591 1/20 0.38
MARK3 P27448 1/20 0.38
FLT3 P36888 1/20 0.38
MAP4K2 Q12851 1/20 0.38
PKN2 Q16513 1/20 0.38
CDC42BPA Q5VT25 1/20 0.38
SLK Q9H2G2 1/20 0.38
IRAK4 Q9NWZ3 1/20 0.38
PIM2 Q9P1W9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL701463 0.76 ALDH1A1 (0.55) ALDH1A1HTTSMN1; SMN2POLBLMNA
SCHEMBL10968043 0.76 ALDH1A1 (0.55) ALDH1A1HTTSMN1; SMN2POLBLMNA
SCHEMBL95810 0.75 BCAT2 (0.40) ALDH1A1HTTSMN1; SMN2LMNA
SCHEMBL23057072 0.74 ALDH1A1 (0.53) ALDH1A1HTTSMN1; SMN2POLBLMNA
SCHEMBL2229460 0.74 PGR (0.54) ALDH1A1HTTSMN1; SMN2POLBKCNJ6
SCHEMBL30908488 0.74 GAA (0.58) ALDH1A1HTTSMN1; SMN2POLBLMNA
SCHEMBL14894969 0.74 ALDH1A1 (0.53) ALDH1A1HTTSMN1; SMN2POLBLMNA
SCHEMBL1439407 0.74 GAA (0.58) ALDH1A1HTTSMN1; SMN2POLBLMNA
SCHEMBL7234031 0.74 ALDH1A1 (0.53) ALDH1A1HTTSMN1; SMN2POLBLMNA
SCHEMBL29558069 0.74 CA1 (0.56) ALDH1A1HTTSMN1; SMN2POLBLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6054469-A Substituted tetrahydropyridine derivatives acting on 5-HT receptors MERCK SHARP & DOHME LTD. (GB) 2000-04-25 US disclosed
US-6048878-A Substituted piperidine derivatives as selective agonists of 5-HT receptors MERCK SHARP & DOHME LTD. (GB) 2000-04-11 US disclosed
EP-0862568-A1 SUBSTITUTED PIPERIDINE DERIVATIVES AS SELECTIVE AGONISTS OF 5-HT RECEPTORS MERCK SHARP & DOHME LTD. (GB) 1998-09-09 EP disclosed
WO-1997018204-A1 SUBSTITUTED TETRAHYDROPYRIDINE DERIVATIVES ACTING ON 5-HT RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 1997-05-22 WO disclosed
WO-1997018202-A1 SUBSTITUTED PIPERIDINE DERIVATIVES AS SELECTIVE AGONISTS OF 5-HT RECEPTORS MERCK SHARP & DOHME LIMITED (GB) 1997-05-22 WO disclosed