SCHEMBL8074863

SCHEMBL8074863

CCc1ccc(C(O)c2ccc(F)c(F)c2)cc1CC

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.44
CES1 P23141 2/20 0.44
PDPK1 O15530 1/20 0.37
MME P08473 1/20 0.36
SHBG P04278 1/20 0.36
ADRB1 P08588 1/20 0.35
ADRA2A P08913 1/20 0.35
ADRB3 P13945 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
KCNQ2 O43526 1/20 0.34
AKR1C3 P42330 2/20 0.33
AKR1C2 P52895 2/20 0.33
ADAM17 P78536 1/20 0.33
HPGD P15428 1/20 0.33
TSHR P16473 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8064216 0.84 NR3C1 (0.40)
SCHEMBL8078157 0.83 CES2 (0.37) CES2CES1ADRB3
SCHEMBL30903827 0.81 CES2 (0.53) CES2CES1PDPK1MMESHBG
SCHEMBL3897101 0.81 CES2 (0.53) CES2CES1PDPK1MMESHBG
SCHEMBL8077682 0.80 LMNA (0.41) CES2CES1SHBGADRB3AKR1C3
SCHEMBL8077592 0.80 CES2 (0.44) CES2CES1
SCHEMBL8074822 0.79 SLC6A2 (0.43) CES2CES1
SCHEMBL2755399 0.79 LMNA (0.44) ADRB3
SCHEMBL8064222 0.79 KCNH2 (0.40)
SCHEMBL8064415 0.78 CYP3A4 (0.42) CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166072-A Amino acid derivatives ALLELIX NEUROSCIENCE, INC. (CA) 2000-12-26 US disclosed
WO-1999034790-A1 GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-07-15 WO disclosed