SCHEMBL8077682

SCHEMBL8077682

CCc1ccc(C(O)c2c(F)cccc2F)cc1CC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
SLC6A2 P23975 5/20 0.33
SLC6A4 P31645 5/20 0.33
CYP3A4 P08684 4/20 0.33
CYP2D6 P10635 4/20 0.33
SLC6A3 Q01959 4/20 0.33
KCNH2 Q12809 4/20 0.33
ALDH1A1 P00352 1/20 0.32
ADRB3 P13945 1/20 0.32
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
RECQL P46063 1/20 0.31
AKR1C3 P42330 1/20 0.31
AKR1C2 P52895 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8074822 0.83 SLC6A2 (0.43) LMNACES2CES1SLC6A2SLC6A4
SCHEMBL8077592 0.81 CES2 (0.44) LMNASMN1; SMN2L3MBTL1CES2CES1
SCHEMBL8074863 0.80 CES2 (0.44) CES2CES1ADRB3AKR1C3AKR1C2
SCHEMBL8064216 0.78 NR3C1 (0.40) LMNAALDH1A1
SCHEMBL8078157 0.77 CES2 (0.37) LMNACES2CES1SLC6A2SLC6A4
SCHEMBL2755399 0.76 LMNA (0.44) LMNASMN1; SMN2L3MBTL1ADRB3
SCHEMBL8064415 0.75 CYP3A4 (0.42) SMN1; SMN2CES2CES1SLC6A2SLC6A4
SCHEMBL8064222 0.73 KCNH2 (0.40) SLC6A2SLC6A4CYP3A4SLC6A3KCNH2
SCHEMBL21830989 0.71 ATM (0.44) CES2CES1ALDH1A1
SCHEMBL8065843 0.71 PDE2A (0.57) SLC6A2SLC6A4CYP3A4SLC6A3AKR1C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166072-A Amino acid derivatives ALLELIX NEUROSCIENCE, INC. (CA) 2000-12-26 US disclosed
WO-1999034790-A1 GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-07-15 WO disclosed