SCHEMBL8074822

SCHEMBL8074822

CCc1ccc(C(O)c2ccccc2F)cc1CC

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SLC6A2 P23975 6/20 0.43
SLC6A4 P31645 6/20 0.43
SLC6A3 Q01959 6/20 0.43
CYP3A4 P08684 6/20 0.43
CYP2D6 P10635 5/20 0.43
KCNH2 Q12809 5/20 0.43
BRD4 O60885 1/20 0.39
CES2 O00748 1/20 0.38
CES1 P23141 1/20 0.38
GAA P10253 1/20 0.35
CNR2 P34972 1/20 0.34
ALDH1A1 P00352 1/20 0.34
LMNA P02545 1/20 0.34
MC4R P32245 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8064415 0.83 CYP3A4 (0.42) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL8077682 0.83 LMNA (0.41) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6
SCHEMBL8064222 0.81 KCNH2 (0.40) SLC6A2SLC6A4SLC6A3CYP3A4KCNH2
SCHEMBL8074863 0.79 CES2 (0.44) CES2CES1
SCHEMBL8072598 0.79 MTNR1B (0.42) LMNA
SCHEMBL8065843 0.79 PDE2A (0.57) SLC6A2SLC6A4SLC6A3CYP3A4
SCHEMBL2755399 0.78 LMNA (0.44) LMNA
SCHEMBL8064216 0.77 NR3C1 (0.40) BRD4ALDH1A1LMNA
SCHEMBL8077592 0.76 CES2 (0.44) SLC6A2SLC6A4BRD4CES2CES1
SCHEMBL8078157 0.76 CES2 (0.37) SLC6A2SLC6A4SLC6A3CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6166072-A Amino acid derivatives ALLELIX NEUROSCIENCE, INC. (CA) 2000-12-26 US disclosed
WO-1999034790-A1 GLYCINE TRANSPORT INHIBITORS ALLELIX NEUROSCIENCE, INC. (US) 1999-07-15 WO disclosed