SCHEMBL808081

SCHEMBL808081

C=C(CN1CCOCC1)C(=O)N1CC[C@H](Nc2cc(CN3C[C@@H](C)O[C@@H](C)C3)cc(Nc3nc4cccnc4s3)n2)C1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.54
RORC P51449 1/20 0.39
DHODH Q02127 1/20 0.39
HCK P08631 7/20 0.38
BTK Q06187 7/20 0.38
SSTR5 P35346 1/20 0.38
LCK P06239 2/20 0.37
AURKB Q96GD4 1/20 0.37
MLNR O43193 2/20 0.32
PIK3CD O00329 1/20 0.32
PIK3R2 O00459 1/20 0.32
PIK3CA P42336 1/20 0.32
PIK3CB P42338 1/20 0.32
PIK3CG P48736 1/20 0.32
PIK3R5 Q8WYR1 1/20 0.32
PIK3R3 Q92569 1/20 0.32
CNR1 P21554 1/20 0.31
CNR2 P34972 1/20 0.31
LTA4H P09960 1/20 0.31
TBK1 Q9UHD2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807946 0.90 ITK (0.58) ITKRORCDHODHHCKBTK
SCHEMBL807743 0.87 ITK (0.57) ITKRORCDHODHHCKBTK
SCHEMBL808093 0.84 ITK (0.61) ITKRORCDHODHHCKBTK
SCHEMBL807803 0.83 ITK (0.58) ITKRORCDHODHHCKBTK
SCHEMBL10285825 0.82 ITK (0.58) ITKRORCDHODHHCKBTK
SCHEMBL807926 0.81 ITK (0.59) ITKRORCDHODHHCKBTK
SCHEMBL2395616 0.80 ITK (0.56) ITKRORCDHODHBTKSSTR5
SCHEMBL808096 0.80 ITK (0.51) ITKRORCDHODHHCKBTK
SCHEMBL807541 0.79 ITK (0.55) ITKRORCDHODHSSTR5LCK
SCHEMBL807540 0.77 ITK (0.46) ITKRORCDHODHSSTR5LCK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed