SCHEMBL808096

SCHEMBL808096

C[C@@H]1CN(Cc2cc(Nc3nc4cccnc4s3)nc(NC3CCCN(C(=O)CCCN(C)C)C3)c2)C[C@H](C)O1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ITK Q08881 2/20 0.51
RORC P51449 1/20 0.41
DHODH Q02127 1/20 0.41
LCK P06239 1/20 0.37
AURKB Q96GD4 1/20 0.37
BTK Q06187 7/20 0.36
HCK P08631 5/20 0.36
SSTR5 P35346 1/20 0.36
JAK2 O60674 2/20 0.33
JAK3 P52333 2/20 0.33
GFER P55789 1/20 0.33
JAK1 P23458 1/20 0.33
BCHE P06276 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807946 0.83 ITK (0.58) ITKRORCDHODHLCKAURKB
SCHEMBL10285825 0.83 ITK (0.58) ITKRORCDHODHLCKAURKB
SCHEMBL807743 0.83 ITK (0.57) ITKRORCDHODHLCKAURKB
SCHEMBL808093 0.83 ITK (0.61) ITKRORCDHODHLCKAURKB
SCHEMBL807803 0.82 ITK (0.58) ITKRORCDHODHLCKAURKB
SCHEMBL2395616 0.80 ITK (0.56) ITKRORCDHODHLCKAURKB
SCHEMBL808081 0.80 ITK (0.54) ITKRORCDHODHLCKAURKB
SCHEMBL807540 0.79 ITK (0.46) ITKRORCDHODHLCKAURKB
SCHEMBL22374670 0.75 ITK (0.71) ITKRORCDHODHLCKAURKB
SCHEMBL807926 0.73 ITK (0.59) ITKRORCDHODHLCKAURKB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035055-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-22 WO disclosed