SCHEMBL808024

SCHEMBL808024

C=C(/N=C(N)\N=C(/N)c1noc(N2CCCCC2)n1)N(C)c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TSHR P16473 4/20 0.37
ALOX15 P16050 2/20 0.37
TP53 P04637 1/20 0.37
SIGMAR1 Q99720 1/20 0.34
LMNA P02545 3/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ELANE P08246 1/20 0.30
RAB9A P51151 1/20 0.30
USP2 O75604 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL808032 0.88 DHFR (0.34) SIGMAR1
SCHEMBL808343 0.87 SCD (0.34) SIGMAR1
SCHEMBL808232 0.85 CNR2 (0.32) SIGMAR1
SCHEMBL808046 0.82 GAA (0.31)
SCHEMBL808026 0.77
SCHEMBL808333 0.75 NPC1 (0.37) SIGMAR1SMN1; SMN2RAB9A
SCHEMBL807920 0.75 SIGMAR1 (0.33) SIGMAR1
SCHEMBL807956 0.74 PRCP (0.35) MAPT
SCHEMBL808229 0.74 SIGMAR1 (0.32) SIGMAR1
SCHEMBL808221 0.74 SIGMAR1 (0.32) SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed