SCHEMBL808236

SCHEMBL808236

C=C(/N=C(N)\N=C(/N)c1noc(-c2ccc(C(=O)NC3CC3)nc2)n1)N(C)c1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.39
USP30 Q70CQ3 1/20 0.35
HDAC1 Q13547 2/20 0.34
HDAC6 Q9UBN7 2/20 0.34
GABRA1 P14867 4/20 0.34
ACKR3 P25106 1/20 0.34
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
S1PR1 P21453 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
PRKAA2 P54646 2/20 0.33
PRKAB2 O43741 1/20 0.33
PRKAG1 P54619 1/20 0.33
PRKAA1 Q13131 1/20 0.33
PRKAG3 Q9UGI9 1/20 0.33
PRKAG2 Q9UGJ0 1/20 0.33
PRKAB1 Q9Y478 1/20 0.33
MLLT1 Q03111 1/20 0.33
KDM1A O60341 1/20 0.32
TGFBR1 P36897 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL808237 0.89 HIF1A (0.39) USP30GABRA1MLLT1
SCHEMBL10287152 0.88 HDAC6 (0.34) HDAC1HDAC6NPC1RAB9AHDAC8
SCHEMBL808234 0.87 HDAC6 (0.34) HDAC1HDAC6NPC1RAB9AHDAC8
SCHEMBL10287197 0.85 CPT2 (0.33) TSHRACKR3NPC1RAB9AKDM1A
SCHEMBL10286912 0.85 GABRA1 (0.36) HDAC1HDAC6GABRA1HDAC8TGFBR1
SCHEMBL808241 0.83 HDAC6 (0.33) HDAC1HDAC6HDAC8
SCHEMBL10287297 0.79 ACACB (0.36)
SCHEMBL807936 0.79 KCNH2 (0.32) USP30
SCHEMBL808331 0.79 KCNH2 (0.32) TSHRUSP30S1PR1
SCHEMBL808333 0.79 NPC1 (0.37) HDAC1HDAC6NPC1RAB9AHDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed