SCHEMBL807936

SCHEMBL807936

C=C(/N=C(N)\N=C(/N)c1noc(-c2ccc(OC3CCC3)nc2)n1)N(C)c1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.32
MCHR1 Q99705 1/20 0.32
SCN9A Q15858 1/20 0.30
GABRA5 P31644 1/20 0.30
USP30 Q70CQ3 1/20 0.30
DGAT1 O75907 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL808331 0.98 KCNH2 (0.32) KCNH2MCHR1SCN9AGABRA5USP30
SCHEMBL807787 0.94 SCN9A (0.37) SCN9AGABRA5
SCHEMBL808238 0.90 TDO2 (0.36) KCNH2MCHR1USP30
SCHEMBL10287297 0.87 ACACB (0.36) GABRA5
SCHEMBL10287197 0.85 CPT2 (0.33) KCNH2MCHR1
SCHEMBL807937 0.83 GABRA5 (0.34) GABRA5
SCHEMBL808332 0.82 GABRA5 (0.34) KCNH2SCN9AGABRA5
SCHEMBL10287152 0.81 HDAC6 (0.34)
SCHEMBL808159 0.80 ACHE (0.31)
SCHEMBL808234 0.80 HDAC6 (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed