SCHEMBL808331

SCHEMBL808331

C=C(/N=C(N)\N=C(/N)c1noc(-c2ccc(OC3CCCCC3)nc2)n1)N(C)c1ccccc1

nearest known ligand 0.32

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.32
MCHR1 Q99705 1/20 0.32
POLB P06746 1/20 0.31
CASP3 P42574 1/20 0.31
SENP7 Q9BQF6 1/20 0.31
SENP6 Q9GZR1 1/20 0.31
S1PR1 P21453 1/20 0.30
S1PR3 Q99500 1/20 0.30
CPT2 P23786 1/20 0.30
CPT1A P50416 1/20 0.30
TSHR P16473 1/20 0.30
SCN9A Q15858 1/20 0.30
GABRA5 P31644 1/20 0.30
USP30 Q70CQ3 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807936 0.98 KCNH2 (0.32) KCNH2MCHR1SCN9AGABRA5USP30
SCHEMBL807787 0.93 SCN9A (0.37) SCN9AGABRA5
SCHEMBL808238 0.89 TDO2 (0.36) KCNH2MCHR1USP30
SCHEMBL10287297 0.86 ACACB (0.36) GABRA5
SCHEMBL10287197 0.86 CPT2 (0.33) KCNH2MCHR1CPT2CPT1ATSHR
SCHEMBL807937 0.82 GABRA5 (0.34) GABRA5
SCHEMBL10287152 0.80 HDAC6 (0.34) POLB
SCHEMBL808234 0.79 HDAC6 (0.34)
SCHEMBL10287187 0.78 ALDH1A1 (0.45) S1PR1
SCHEMBL808333 0.77 NPC1 (0.37) POLBCASP3SENP7SENP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed