SCHEMBL808241

SCHEMBL808241

C=C(/N=C(N)\N=C(/N)c1noc(-c2ccc(C(=O)OC(C)C)nc2)n1)N(C)c1ccccc1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 3/20 0.33
HDAC1 Q13547 2/20 0.33
KMT2A Q03164 2/20 0.32
HDAC8 Q9BY41 2/20 0.32
ALOX5AP P20292 1/20 0.31
HDAC4 P56524 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10287152 0.89 HDAC6 (0.34) HDAC6HDAC1HDAC8HDAC4
SCHEMBL808234 0.88 HDAC6 (0.34) HDAC6HDAC1HDAC8HDAC4
SCHEMBL10287197 0.87 CPT2 (0.33) ALOX5AP
SCHEMBL808236 0.83 TSHR (0.39) HDAC6HDAC1HDAC8
SCHEMBL10286912 0.81 GABRA1 (0.36) HDAC6HDAC1HDAC8HDAC4
SCHEMBL808237 0.81 HIF1A (0.39)
SCHEMBL808161 0.78 HDAC4 (0.32) HDAC6HDAC8HDAC4
SCHEMBL807937 0.78 GABRA5 (0.34)
SCHEMBL808333 0.78 NPC1 (0.37) HDAC6HDAC1KMT2AHDAC8HDAC4
SCHEMBL10287297 0.77 ACACB (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed