SCHEMBL808238

SCHEMBL808238

C=C(/N=C(N)\N=C(/N)c1noc(-c2ccc(OC3CCN(C)C3)nc2)n1)N(C)c1ccccc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 1/20 0.36
ATM Q13315 1/20 0.33
ATR Q13535 1/20 0.33
CHRM4 P08173 1/20 0.33
CHRM5 P08912 1/20 0.33
CHRM1 P11229 1/20 0.33
CHRM3 P20309 1/20 0.33
USP30 Q70CQ3 1/20 0.32
KCNH2 Q12809 1/20 0.32
MCHR1 Q99705 1/20 0.32
ACKR3 P25106 1/20 0.31
PIK3CD O00329 1/20 0.31
NOS3 P29474 1/20 0.31
NOS1 P29475 1/20 0.31
NOS2 P35228 1/20 0.31
PIK3CA P42336 1/20 0.31
HDAC1 Q13547 1/20 0.30
HDAC8 Q9BY41 1/20 0.30
HDAC6 Q9UBN7 1/20 0.30
USP7 Q93009 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL807936 0.90 KCNH2 (0.32) USP30KCNH2MCHR1
SCHEMBL808331 0.89 KCNH2 (0.32) USP30KCNH2MCHR1
SCHEMBL10287297 0.85 ACACB (0.36)
SCHEMBL807937 0.80 GABRA5 (0.34)
SCHEMBL10287197 0.79 CPT2 (0.33) KCNH2MCHR1ACKR3
SCHEMBL10287152 0.77 HDAC6 (0.34) HDAC1HDAC8HDAC6
SCHEMBL808234 0.77 HDAC6 (0.34) HDAC1HDAC8HDAC6
SCHEMBL808237 0.76 HIF1A (0.39) USP30
SCHEMBL808333 0.75 NPC1 (0.37) HDAC1HDAC8HDAC6
SCHEMBL808241 0.74 HDAC6 (0.33) HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012035023-A1 TRIAZINE-OXADIAZOLES NOVARTIS AG (CH) 2012-03-22 WO disclosed